{"id":4345,"date":"2013-10-13T17:58:08","date_gmt":"2013-10-13T15:58:08","guid":{"rendered":"https:\/\/dixitciencia.com\/2013\/10\/13\/reciclando-farmacos-del-corazon-al-cancer\/"},"modified":"2017-05-02T07:27:07","modified_gmt":"2017-05-02T07:27:07","slug":"reciclant-farmacs-del-cor-al-cancer","status":"publish","type":"post","link":"https:\/\/dixitciencia.com\/ca\/2013\/10\/13\/reciclant-farmacs-del-cor-al-cancer\/","title":{"rendered":"Reciclant f\u00e0rmacs: del cor al c\u00e0ncer"},"content":{"rendered":"<p style=\"text-align: justify;\">\u2022 En la recerca de f\u00e0rmacs contra el c\u00e0ncer (com en molts altres camps de la ci\u00e8ncia) la teoria no sempre precedeix la pr\u00e0ctica. Sovint,\u00a0<strong>en una obligada lli\u00e7\u00f3 d\u2019humilitat a priori,<\/strong>\u00a0les primeres passes s\u00f3n pals de cec, una mena de r\u00e0fegues de metralleta buscant algun tret que faci diana. La qual cosa no deixa de ser \u00fatil. Un exemple \u00e9s l\u2019anomenat\u00a0<a title=\"\" href=\"http:\/\/www.nature.com\/nrc\/journal\/v6\/n10\/full\/nrc1951.html\" target=\"_blank\" rel=\"noopener noreferrer\">NCI-60<\/a>, un projecte que va comen\u00e7ar als 80 i que ha analitzat m\u00e9s de 100.000 compostos, ja siguin sint\u00e8tics o naturals, provinents dels m\u00e9s variats racons del planeta (de plantes, animals marins, microorganismes). En ess\u00e8ncia, del que es tracta \u00e9s d\u2019estudiar si alguna d\u2019aquestes subst\u00e0ncies \u00e9s capa\u00e7 d\u2019aturar el creixement d\u2019algun dels 60 tumors que es van seleccionar. Si alguna d\u2019elles demostra tenir un efecte, s\u2019inicia un complex proc\u00e9s que, en alguns casos, acaba arribant als hospitals. Per\u00f2:<\/p>\n<p style=\"text-align: justify;\">&#8211; Tan sols un de cada 5.000 o 10.000 compostos que es proven acaben sent utilitzats.<\/p>\n<p style=\"text-align: justify;\">&#8211; \u00danicament un 5% dels que es comencen provant en humans arriben a ser finalment aprovats, i arribats a aquest punt<\/p>\n<p style=\"text-align: justify;\">&#8211; La mitjana del proc\u00e9s \u00e9s d\u2019uns 13 anys, amb uns costos considerables.<\/p>\n<p style=\"text-align: justify;\">\u2022 Una altra opci\u00f3, que implica una mica menys d\u2019humilitat ja que concedeix un major paper al cient\u00edfic, \u00e9s aprofitar part del que ja \u00e9s conegut: \u00e9s estrany el f\u00e0rmac que nom\u00e9s actua sobre un \u00fanic punt de la c\u00e8l\u00b7lula. En general la naturalesa, i el que fem per controlar-la, \u00e9s una mica m\u00e9s bruta en el seu <a href=\"https:\/\/dixitciencia.com\/wp-content\/uploads\/6a01347ff0d110970c01676267475c970b-500wi3-1.jpg\" class=\"mfp-image\"><img loading=\"lazy\" decoding=\"async\" class=\"alignleft size-medium wp-image-1608 lazyload\" style=\"margin: 8px 14px;\" title=\"6a01347ff0d110970c01676267475c970b-500wi\" src=\"data:image\/gif;base64,R0lGODlhAQABAAAAACH5BAEKAAEALAAAAAABAAEAAAICTAEAOw==\" data-src=\"https:\/\/dixitciencia.com\/wp-content\/uploads\/6a01347ff0d110970c01676267475c970b-500wi3-300x199-1.jpg\" alt=\"\" width=\"300\" height=\"199\" \/><\/a>comportament. \u00c9s possible, per tant, que <strong>f\u00e0rmacs aprovats per a unes malalties puguin ser beneficiosos en d\u2019altres<\/strong>. Si \u00e9s aix\u00ed, ens estalviar\u00edem una gran part del cam\u00ed: coneixer\u00edem les dosis a emprar, les possibles contraindicacions, els efectes secundaris. <strong>Comen\u00e7ar\u00edem la cursa a la meitat<\/strong>.<\/p>\n<p style=\"text-align: justify;\">Aix\u00f2 \u00e9s el que han fet\u00a0<a title=\"\" href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/22814852\" target=\"_blank\" rel=\"noopener noreferrer\">uns investigadors<\/a>\u00a0als Estats Units. Limitar els pals de cec de dues maneres: d\u2019una banda van aprofitar el coneixement que alguns tractaments contra el c\u00e0ncer s\u00f3n efica\u00e7os perqu\u00e8 \u201censenyen\u201d al sistema immunitari a atacar el tumor. D\u2019altra, van buscar aquests senyals despr\u00e9s de provar poc m\u00e9s de 1.000 f\u00e0rmacs, tots ells ja aprovats per a diferents malalties. Els resultats?<\/p>\n<p style=\"text-align: justify;\">Entre els f\u00e0rmacs m\u00e9s efica\u00e7os estaven aquells que ja s\u2019usaven amb aquest prop\u00f2sit. Per\u00f2 entre ells es va colar un de particularment popular i que no tenia res a veure a priori amb el c\u00e0ncer: era la <strong>digoxina<\/strong>, un medicament \u00e0mpliament utilitzat per tractar les ar\u00edtmies card\u00edaques. Despr\u00e9s van analitzar les dades hospital\u00e0ries que tenien des dels anys 80: aquells pacients amb c\u00e0ncer que tamb\u00e9 patien ar\u00edtmies i estaven sent tractats amb digoxina sobrevivien m\u00e9s temps que no pas la resta.<\/p>\n<p style=\"text-align: justify;\">Falten els estudis definitius, no comenceu a prendre digoxina (f\u00e0rmac delicat, d\u2019altra banda), per\u00f2 no \u00e9s desgavellat pensar en aquest paradoxal reciclatge.<\/p>\n<p style=\"text-align: justify;\"><strong>\u00b7<\/strong> I encara hi ha m\u00e9s opcions, cada vegada exigint una menor quota d\u2019humilitat:<\/p>\n<p style=\"text-align: justify;\">El fet que gaireb\u00e9 cap medicament actu\u00ef \u00fanicament sobre un rac\u00f3 cel\u00b7lular \u00e9s la principal ra\u00f3 que hi hagi <strong>efectes secundaris<\/strong>. Per\u00f2 <strong>all\u00f2 que perjudica alg\u00fa \u00e9s possible que sigui el que un altre necessiti<\/strong>. Per exemple:<\/p>\n<p style=\"text-align: justify;\">&#8211; La <strong>talidomida<\/strong> \u00e9s un f\u00e0rmac que es va usar al voltant dels anys 60 per disminuir les n\u00e0usees de les embarassades. No obstant, es va veure que provocava greus malformacions en els nens, motiu pel qual va ser retirat del mercat. Un dels mecanismes proposats era que alterava la formaci\u00f3 de vasos sanguinis, i aquest efecte (entre altres) \u00e9s el que ara permet que es faci servir en el tractament de tumors com el mieloma m\u00faltiple.<\/p>\n<p style=\"text-align: justify;\">Aquest \u00e9s nom\u00e9s un exemple. Ja hi ha equips de\u00a0<strong><a title=\"\" href=\"http:\/\/www.usc.es\/biofarma\/en\/index.htm\" target=\"_blank\" rel=\"noopener noreferrer\">rastrejadors<\/a>\u00a0<\/strong>d\u2019efectes secundaris. I no nom\u00e9s buscant f\u00e0rmacs contra el c\u00e0ncer, sin\u00f3 tamb\u00e9 pel tractament de malalties neurol\u00f2giques, la diabetis o l\u2019ampli llistat de les conegudes com a malalties rares.<\/p>\n<p style=\"text-align: justify;\">(Per cert, la <strong>Viagra<\/strong> va ser desenvolupada com un medicament contra la hipertensi\u00f3. Les ereccions que provocava van ser considerades en principi com un efecte secundari.)<\/p>\n<p style=\"text-align: justify;\">Si tantes vegades les modes han demostrat ser c\u00edcliques, haurem de donar una oportunitat al\u00a0<em>vintage.<\/em><\/p>\n<p style=\"text-align: justify;\">*<\/p>\n<p style=\"text-align: justify;\">Aquest article va ser publicat el 01\/10\/2013 al diari digital <a href=\"http:\/\/www.50x7.com\/reciclant-farmacs\/\" target=\"_blank\" rel=\"noopener noreferrer\">50&#215;7.com<\/a><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Perqu\u00e8 la Viagra \u00e9s \u00fatil gr\u00e0cies a un efecte secundari. Perqu\u00e8 hi ha drogues per al cor que semblen ser efica\u00e7os contra el c\u00e0ncer. Perqu\u00e8 el reciclatge en l&#8217;\u00fas de f\u00e0rmacs ens permet estalviar costos i comen\u00e7ar la cursa a la meitat.<\/p>\n","protected":false},"author":2,"featured_media":4348,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"jetpack_post_was_ever_published":false,"_jetpack_newsletter_access":"","_jetpack_dont_email_post_to_subs":false,"_jetpack_newsletter_tier_id":0,"_jetpack_memberships_contains_paywalled_content":false,"_jetpack_memberships_contains_paid_content":false,"footnotes":""},"categories":[838,813],"tags":[1004,1005,1006,1007,822,1008,1009,1010,1011,1012],"thb-sponsors":[],"class_list":["post-4345","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-biomedicina-i-salut","category-general-ca","tag-cancer-ca","tag-digoxina-ca","tag-farmacos-ca","tag-farmacs-ca","tag-investigacion-ca","tag-medicamentos-ca","tag-reciclaje-ca","tag-reciclatge-ca","tag-reposicionamiento-ca","tag-viagra-ca"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.0 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Reciclant f\u00e0rmacs: del cor al c\u00e0ncer - Dixit<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/dixitciencia.com\/2013\/10\/13\/reciclando-farmacos-del-corazon-al-cancer\/\" \/>\n<meta property=\"og:locale\" content=\"ca_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Reciclant f\u00e0rmacs: del cor al c\u00e0ncer - Dixit\" \/>\n<meta property=\"og:description\" content=\"Perqu\u00e8 la Viagra \u00e9s \u00fatil gr\u00e0cies a un efecte secundari. 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